夏霖, 倪沛洲, 宋武, 刘国卿, 钱家庆, 李蓓, 桂冠华. 苯氧烷胺类化合物的合成及其抗高血压活性J. 药学学报, 1990, 25(2): 150-153.
引用本文: 夏霖, 倪沛洲, 宋武, 刘国卿, 钱家庆, 李蓓, 桂冠华. 苯氧烷胺类化合物的合成及其抗高血压活性J. 药学学报, 1990, 25(2): 150-153.
L Xia, PZ Ni, W Song, GQ Liu, JQ Qian, P Li , FH Du, . SYNTHESIS AND ANTIHYPERTENSIVE ACTIVITY OF SOME PHENOXYALKYLAMINE COMPOUNDSJ. Acta Pharmaceutica Sinica, 1990, 25(2): 150-153.
Citation: L Xia, PZ Ni, W Song, GQ Liu, JQ Qian, P Li , FH Du, . SYNTHESIS AND ANTIHYPERTENSIVE ACTIVITY OF SOME PHENOXYALKYLAMINE COMPOUNDSJ. Acta Pharmaceutica Sinica, 1990, 25(2): 150-153.

苯氧烷胺类化合物的合成及其抗高血压活性

SYNTHESIS AND ANTIHYPERTENSIVE ACTIVITY OF SOME PHENOXYALKYLAMINE COMPOUNDS

  • Abstract: Nine new compounds were synthesized and tested for their α-adrenoceptor affinity and antihypertensive activity together with 5 other previously reported compounds(1). Compounds Ⅰ, Ⅱa, Ⅱb and Ⅲa showed high α-adrenoceptor affinity and strong antihypertensive activity.

     

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